SCHEMBL6965142

SCHEMBL6965142

Nc1cc(Sc2cccc3cnccc23)c(Cl)cc1[N+](=O)[O-]

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 12/20 0.47
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
ALDH1A1 P00352 1/20 0.42
SLC6A4 P31645 1/20 0.41
MAPT P10636 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
GAA P10253 1/20 0.41
MAPK1 P28482 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.39
PSMD14 O00487 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972315 0.91 LMNA (0.46) PDE7AMEN1KMT2ALMNACYP1A2
SCHEMBL6958271 0.87 LMNA (0.42) PDE7AMEN1KMT2ALMNACYP1A2
SCHEMBL6965245 0.87 LMNA (0.42) PDE7AMEN1KMT2ALMNACYP1A2
SCHEMBL6963335 0.86 LMNA (0.46) PDE7AMEN1KMT2ALMNACYP1A2
SCHEMBL6962927 0.84 LMNA (0.51) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6958268 0.84 LMNA (0.42) PDE7AMEN1KMT2ALMNACYP1A2
SCHEMBL6966094 0.84 LMNA (0.43) PDE7AMEN1KMT2ALMNACYP1A2
SCHEMBL6966276 0.84 MAPT (0.42) PDE7AMEN1KMT2ALMNACYP1A2
SCHEMBL6968103 0.81 MAPT (0.48) PDE7AMEN1KMT2ALMNACYP1A2
SCHEMBL6973656 0.81 PDE7A (0.60) PDE7AMEN1KMT2ALMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed