SCHEMBL6965417

SCHEMBL6965417

CC(C)c1c(Sc2ccccc2)nc(COC(N)=O)n1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.37
TOP2A P11388 2/20 0.36
TOP2B Q02880 2/20 0.36
EPHX1 P07099 1/20 0.36
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CYP1A2 P05177 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
CXCL12 P48061 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
CYP2D6 P10635 2/20 0.33
MAPT P10636 2/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967031 0.89 CYP1A2 (0.44) TOP2ATOP2BALDH1A1POLBTDP1
SCHEMBL6969756 0.87 ALOX12 (0.40) LMNAALDH1A1POLBCYP1A2CYP2C9
SCHEMBL7084947 0.87 EPHX1 (0.37) LMNAEPHX1ALDH1A1L3MBTL1MAPT
SCHEMBL6971287 0.86 ALDH1A1 (0.36) LMNATOP2ATOP2BEPHX1ALDH1A1
SCHEMBL6969923 0.85 LMNA (0.36) LMNAEPHX1CYP1A2CYP2C9CYP2C19
SCHEMBL6975484 0.84 LMNA (0.36) LMNA
SCHEMBL7082337 0.84 LMNA (0.36) LMNACYP1A2CYP2C9CYP2C19L3MBTL1
SCHEMBL6974900 0.84 LMNA (0.42) LMNAALDH1A1POLBTDP1CYP2C9
SCHEMBL6969941 0.81 CYP1A2 (0.39) LMNATOP2ATOP2BEPHX1CYP1A2
SCHEMBL6973086 0.81 PIM1 (0.36) LMNATOP2ATOP2BALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed