SCHEMBL6965778

SCHEMBL6965778

c1ccc(NCCOc2ccccn2)cc1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
F2 P00734 5/20 0.46
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45
HTR1A P08908 3/20 0.42
ADRA1D P25100 3/20 0.42
ADRA1A P35348 3/20 0.42
ADRA1B P35368 3/20 0.42
METAP1 P53582 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
AURKA O14965 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29236607 0.84 ALDH1A1 (0.54) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL4190714 0.78 KDM4E (0.50) ALDH1A1METAP1NPC1RAB9AL3MBTL1
SCHEMBL2569101 0.78 HTR1B (0.55) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL13940266 0.76 HTR1B (0.56) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL13900538 0.76 DRD4 (0.62) MAOAHTR1AADRA1DADRA1AADRA1B
SCHEMBL1953722 0.76 MTNR1A (0.46) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL8725186 0.75 DRD4 (0.61) F2ALDH1A1MAPTNPC1RAB9A
SCHEMBL15617823 0.75 NPC1 (0.43) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL29969403 0.75 HTR1A (0.45) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL29629169 0.74 HTR1B (0.50) HTR1AADRA1DADRA1AADRA1BNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1021411-B1 BENZAMIDE DERIVATIVES AS THROMBIN INHIBITORS GLAXO GROUP LTD (GB) 2003-03-05 EP disclosed
US-6326386-B1 ANTICOAGULANT GLAXO GROUP LIMITED (GB) 2001-12-04 US disclosed