SCHEMBL6966304

SCHEMBL6966304

C/C=C1\CNCC[C@H]1CCCc1ccnc2ccc(O)cc12

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.34
SLC6A4 P31645 1/20 0.32
MTNR1A P48039 1/20 0.30
MTNR1B P49286 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6966308 1.00 TRPV1 (0.34) TRPV1SLC6A4MTNR1AMTNR1B
SCHEMBL6972322 0.76 DRD3 (0.37)
SCHEMBL6972325 0.76 DRD3 (0.37)
SCHEMBL6978373 0.76 TRPV1 (0.35) TRPV1SLC6A4MTNR1AMTNR1B
SCHEMBL22728221 0.70 TYR (0.51) TRPV1MTNR1AMTNR1B
SCHEMBL23487414 0.67 CYP2D6 (0.34) TRPV1SLC6A4
SCHEMBL8124875 0.66 ENPP1 (0.35) TRPV1
SCHEMBL11338421 0.65 SLC6A4 (0.40) SLC6A4
SCHEMBL18664158 0.65 TRPV1 (0.37) TRPV1SLC6A4MTNR1AMTNR1B
SCHEMBL4075615 0.64 ESR1 (0.54) TRPV1MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051413-B1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2003-06-04 EP disclosed
EP-1051413-A1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2000-11-15 EP disclosed
WO-1999037635-A1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 1999-07-29 WO disclosed