SCHEMBL8124875

SCHEMBL8124875

CC=C(CCCC)CCN1CCC(CCCc2ccnc3ccc(O)cc23)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP1 P22413 1/20 0.35
KCNH2 Q12809 3/20 0.34
CHRM1 P11229 2/20 0.34
DRD2 P14416 2/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
HTR1A P08908 1/20 0.34
CHRM5 P08912 1/20 0.34
ADRA2A P08913 1/20 0.34
ADRA2B P18089 1/20 0.34
CHRM3 P20309 1/20 0.34
DRD4 P21917 1/20 0.34
ADRA1D P25100 1/20 0.34
ADRA1A P35348 1/20 0.34
HRH1 P35367 1/20 0.34
ADRA1B P35368 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
ACHE P22303 2/20 0.33
HTR4 Q13639 2/20 0.33
NMT1 P30419 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972325 0.76 DRD3 (0.37) KCNH2DRD2HTR1ADRD4DRD3
SCHEMBL6972322 0.76 DRD3 (0.37) KCNH2DRD2HTR1ADRD4DRD3
SCHEMBL6975728 0.74 CCR8 (0.56) KCNH2
SCHEMBL6965739 0.74 DRD3 (0.45) DRD2HTR1ADRD4DRD3
SCHEMBL22728221 0.73 TYR (0.51) TRPV1
SCHEMBL8133161 0.71 CCR8 (0.45) KCNH2HTR1AHRH3
SCHEMBL23487414 0.70 CYP2D6 (0.34) ENPP1KCNH2DRD2ADRA2AADRA2B
SCHEMBL11338421 0.68 SLC6A4 (0.40) KCNH2CHRM2HRH3NMT1
SCHEMBL6966304 0.66 TRPV1 (0.34) TRPV1
SCHEMBL6966308 0.66 TRPV1 (0.34) TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051413-A1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2000-11-15 EP disclosed
WO-1999037635-A1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 1999-07-29 WO disclosed