SCHEMBL6966448

SCHEMBL6966448

Nc1ccc(Sc2cccc3cnccc23)nc1N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.53
CYP3A4 P08684 2/20 0.53
CYP2D6 P10635 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
IMPDH2 P12268 4/20 0.43
KDM4E B2RXH2 1/20 0.41
MAPKAPK2 P49137 1/20 0.41
HTT P42858 1/20 0.39
CCR4 P51679 1/20 0.34
AXL P30530 1/20 0.34
EP300 Q09472 1/20 0.34
KAT2B Q92831 1/20 0.34
KAT8 Q9H7Z6 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
PRKD3 O94806 1/20 0.34
TP53 P04637 1/20 0.34
PRKCG P05129 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6961993 0.81 MAPT (0.43) LMNACYP3A4CYP2D6CYP1A2CYP2C9
SCHEMBL6968741 0.79 KDM4E (0.57) LMNACYP3A4CYP2D6CYP1A2CYP2C9
SCHEMBL6958264 0.77 CYP3A4 (0.53) LMNACYP3A4CYP2D6CYP1A2CYP2C9
SCHEMBL6973375 0.75 LMNA (0.54) LMNACYP3A4CYP2D6CYP1A2CYP2C9
SCHEMBL6966830 0.74 KDM4E (0.49) LMNACYP3A4CYP2D6CYP1A2CYP2C9
SCHEMBL6968806 0.73 LMNA (0.51) LMNACYP3A4CYP2D6CYP1A2CYP2C9
SCHEMBL6962927 0.73 LMNA (0.51) LMNACYP3A4CYP2D6CYP1A2CYP2C9
SCHEMBL6973379 0.73 CYP3A4 (0.51) LMNACYP3A4CYP2D6CYP1A2CYP2C9
SCHEMBL8282774 0.73 CYP3A4 (0.58) LMNACYP3A4CYP2D6CYP1A2CYP2C9
SCHEMBL6969782 0.72 LMNA (0.57) LMNAKDM4EHTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed