SCHEMBL6973379

SCHEMBL6973379

Nc1cc(F)c(Sc2cccc3cnccc23)cc1N

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.51
CYP2D6 P10635 2/20 0.51
LMNA P02545 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
IMPDH2 P12268 4/20 0.42
KDM4E B2RXH2 3/20 0.41
MAPKAPK2 P49137 1/20 0.41
MAPT P10636 4/20 0.39
ALDH1A1 P00352 2/20 0.39
HTT P42858 3/20 0.38
ROCK2 O75116 1/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
PRKD3 O94806 1/20 0.36
TP53 P04637 1/20 0.36
PRKCG P05129 1/20 0.36
PRKCB P05771 1/20 0.36
PRKCA P17252 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6958271 0.84 LMNA (0.42) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL6962927 0.83 LMNA (0.51) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL6968806 0.83 LMNA (0.51) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL6968741 0.82 KDM4E (0.57) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL6973375 0.80 LMNA (0.54) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL6958264 0.79 CYP3A4 (0.53) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL6963335 0.78 LMNA (0.46) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL6963265 0.76 HTT (0.47) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL6972315 0.76 LMNA (0.46) CYP3A4CYP2D6LMNACYP1A2CYP2C9
SCHEMBL6965245 0.74 LMNA (0.42) CYP3A4CYP2D6LMNACYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed