SCHEMBL6966536

SCHEMBL6966536

Cc1cc(C)cc(Sc2cnc(C)[nH]2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 1/20 0.37
HRH4 Q9H3N8 1/20 0.37
BAZ2B Q9UIF8 1/20 0.32
NOTUM Q6P988 1/20 0.32
TUBB4A P04350 1/20 0.31
TUBB P07437 1/20 0.31
TUBA3C P0DPH7 1/20 0.31
IDO1 P14902 1/20 0.31
TUBA1B P68363 1/20 0.31
TUBA4A P68366 1/20 0.31
TUBB4B P68371 1/20 0.31
TUBB3 Q13509 1/20 0.31
TUBB2A Q13885 1/20 0.31
TUBB8 Q3ZCM7 1/20 0.31
TUBA3E Q6PEY2 1/20 0.31
TUBA1A Q71U36 1/20 0.31
TUBA1C Q9BQE3 1/20 0.31
TUBB6 Q9BUF5 1/20 0.31
TUBB2B Q9BVA1 1/20 0.31
TUBB1 Q9H4B7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9291589 0.69 HRH4 (0.50) HRH1HRH4FDPS
SCHEMBL3689119 0.68 ALDH1A1 (0.44) NOTUMTUBB4ATUBBTUBA3CIDO1
SCHEMBL9291587 0.68 HRH1 (0.33) HRH1HRH4
SCHEMBL14252153 0.66 ALDH1A1 (0.42) NOTUMTUBB4ATUBBTUBA3CIDO1
SCHEMBL6971477 0.65 HEXA (0.34)
SCHEMBL6966153 0.63 CDK4 (0.30)
SCHEMBL112709 0.59
SCHEMBL19265598 0.58 MLYCD (0.45)
SCHEMBL7187600 0.58 ALDH1A1 (0.63) NOTUMTUBB4ATUBBTUBA3CIDO1
SCHEMBL4032966 0.58 ALDH1A1 (0.44) TUBB4ATUBBTUBA3CIDO1TUBA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed