SCHEMBL6971477

SCHEMBL6971477

CCc1nc(C)[nH]c1Sc1cc(C)cc(C)c1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HEXA P06865 1/20 0.34
HEXB P07686 1/20 0.34
TYMS P04818 1/20 0.32
HTT P42858 1/20 0.30
NOS3 P29474 1/20 0.30
NOS2 P35228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6966153 0.85 CDK4 (0.30)
SCHEMBL8562378 0.80 DHFR (0.45) TYMS
SCHEMBL8349406 0.77 USP2 (0.36)
SCHEMBL8349410 0.71 ACHE (0.33)
SCHEMBL6968923 0.66 HEXA (0.33) HEXAHEXBHTTNOS3NOS2
SCHEMBL6086721 0.65 TYMP (0.37)
SCHEMBL6966536 0.65 HRH1 (0.37)
SCHEMBL3689119 0.63 ALDH1A1 (0.44)
SCHEMBL5851367 0.63
SCHEMBL7086346 0.63 CYP1A2 (0.40) HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0552060-B1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO (JP) 1998-11-18 EP disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed
EP-0700911-A1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO., LTD. (JP) 1996-03-13 EP disclosed
US-5472965-A Useful for treatment of retrovirus infections; less toxic SHIONOGI & CO., LTD. (JP) 1995-12-05 US disclosed
US-5326780-A Acquired immunodeficiency syndrome SHIONOGI & CO., LTD. (JP) 1994-07-05 US disclosed
EP-0552060-A1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO., LTD. (JP) 1993-07-21 EP disclosed