SCHEMBL6966632

SCHEMBL6966632

CC(C)c1nc(COC(=O)NC(=O)CCl)n(Cc2ccccc2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.36
RECQL P46063 1/20 0.34
ENPP2 Q13822 2/20 0.33
CCR1 P32246 1/20 0.33
PPARG P37231 1/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
TOP2A P11388 1/20 0.33
TOP2B Q02880 1/20 0.33
P2RX3 P56373 3/20 0.32
ALDH1A1 P00352 1/20 0.32
KCNJ6 P48051 1/20 0.32
KCNJ5 P48544 1/20 0.32
KCNJ3 P48549 1/20 0.32
MAPK1 P28482 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6965855 0.92 ENPP2 (0.33) ENPP2P2RX3
SCHEMBL6973878 0.92 MEN1 (0.35) ENPP2KMT2AMEN1P2RX3ALDH1A1
SCHEMBL6972332 0.90 FAAH (0.35) ENPP2KMT2AMEN1P2RX3
SCHEMBL6964352 0.87
SCHEMBL6161001 0.86 ENPP2 (0.35) TDP1ENPP2KMT2AMEN1P2RX3
SCHEMBL6967638 0.86 TDP1 (0.39) TDP1RECQLKMT2AMEN1P2RX3
SCHEMBL6962947 0.85
Acetamide SCHEMBL6959979 0.84 TDP1 (0.38) TDP1RECQLKMT2AMEN1ALDH1A1
SCHEMBL6167205 0.83 ENPP2 (0.34) ENPP2KMT2AMEN1P2RX3ALDH1A1
SCHEMBL6961504 0.81 ENPP2 (0.35) ENPP2KMT2AMEN1TOP2ATOP2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP claimed
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed