SCHEMBL6966653

SCHEMBL6966653

CCCCCCn1c(COC(N)=O)nc(C(C)C)c1Sc1cc(C)cc(C)c1

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSSK1B Q9BXA7 1/20 0.32
PSEN1 P49768 2/20 0.32
PSEN2 P49810 2/20 0.32
APH1B Q8WW43 2/20 0.32
NCSTN Q92542 2/20 0.32
APH1A Q96BI3 2/20 0.32
PSENEN Q9NZ42 2/20 0.32
GRK6 P43250 2/20 0.32
SIRT2 Q8IXJ6 3/20 0.31
PLA2G2A P14555 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CNR2 P34972 2/20 0.31
TLR8 Q9NR97 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974730 0.96 ALDH1A1 (0.32) ALDH1A1MAPTHTTSMN1; SMN2
SCHEMBL6960602 0.92 SMN1; SMN2 (0.37) ALDH1A1MAPTHTTSMN1; SMN2
SCHEMBL6969235 0.91 TP53 (0.31) TSSK1BPSEN1PSEN2APH1BNCSTN
SCHEMBL7085912 0.90 TP53 (0.32) TSSK1BPSEN1PSEN2APH1BNCSTN
SCHEMBL6963219 0.90 HSP90B1 (0.37) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6973745 0.90 MEN1 (0.32) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6969825 0.88 LMNA (0.31) MAPT
SCHEMBL7084691 0.86 SMN1; SMN2 (0.32) ALDH1A1SMN1; SMN2
SCHEMBL6974759 0.85 HSP90B1 (0.40) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6974392 0.85 CYP1A2 (0.33) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed