SCHEMBL6973745

SCHEMBL6973745

CCCCCCn1c(COC(N)=O)nc(C(C)C)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.32
HPGD P15428 1/20 0.32
KMT2A Q03164 1/20 0.32
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31
CYP1A2 P05177 2/20 0.31
CYP2C9 P11712 2/20 0.31
CYP2C19 P33261 2/20 0.31
ALDH1A1 P00352 1/20 0.31
CNR2 P34972 1/20 0.30
CYP3A4 P08684 1/20 0.30
ICMT O60725 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974392 0.96 CYP1A2 (0.33) MEN1HPGDKMT2ACYP1A2CYP2C9
SCHEMBL6969451 0.92 MEN1 (0.38) MEN1HPGDKMT2ACYP1A2CYP2C9
SCHEMBL6968457 0.91 GCGR (0.32) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6969613 0.90 PPARG (0.33) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6966653 0.90 TSSK1B (0.32) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6963219 0.89 HSP90B1 (0.37) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6967644 0.88 GLA (0.32) MEN1HPGDKMT2ACYP1A2CYP2C9
SCHEMBL6965378 0.88 LMNA (0.32) CYP1A2CYP2C9CYP2C19ALDH1A1CYP3A4
SCHEMBL6966575 0.87 ALDH1A1 (0.33) MEN1HPGDKMT2ACYP1A2CYP2C9
SCHEMBL6969155 0.86 LMNA (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed