SCHEMBL6968874

SCHEMBL6968874

O=C(c1ccccc1)n1cc(CCC2CCCN2)c2cc(Br)ccc21

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 8/20 0.45
HTR1A P08908 1/20 0.45
HTR1D P28221 1/20 0.45
HTR1B P28222 1/20 0.45
HTR1F P30939 1/20 0.45
HTR7 P34969 1/20 0.45
DYRK1A Q13627 1/20 0.42
MBTD1 Q05BQ5 1/20 0.37
PRPS1 P60891 1/20 0.36
ELANE P08246 2/20 0.36
KRAS P01116 1/20 0.36
KHK P50053 1/20 0.35
SLC6A4 P31645 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6976187 0.81 HTR6 (0.39) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL6968868 0.79 HTR6 (0.50) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL6972524 0.75 HTR6 (0.77) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL6968879 0.74 DYRK1A (0.42) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL6965704 0.73 HTR6 (0.49) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL6967984 0.73 HTR6 (0.49) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL6965707 0.73 HTR6 (0.49) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL6968124 0.72 HTR6 (0.36) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL7006184 0.72 SLC6A4 (0.36) HTR6PRPS1SLC6A4
SCHEMBL8483890 0.71 HTR6 (0.61) HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP disclosed
US-5998438-A SEROTONIN RECEPTOR ANTAGONIST; HEADACHE THERAPY ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1999-12-07 US disclosed
EP-0944595-A1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS Allelix Biopharmaceuticals Inc. (CA) 1999-09-29 EP disclosed
WO-1998023587-A1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS ALLELIX BIOPHARMACEUTICALS INC. (CA) 1998-06-04 WO disclosed