SCHEMBL6969253

SCHEMBL6969253

COCc1nc(Cl)nc(N2CCc3cc(OC)ccc3C2C)c1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 5/20 0.40
DRD2 P14416 3/20 0.37
DRD4 P21917 2/20 0.37
TUBB4A P04350 2/20 0.37
TUBB P07437 2/20 0.37
TUBA3C P0DPH7 2/20 0.37
TUBA1B P68363 2/20 0.37
TUBA4A P68366 2/20 0.37
TUBB4B P68371 2/20 0.37
TUBB3 Q13509 2/20 0.37
TUBB2A Q13885 2/20 0.37
TUBB8 Q3ZCM7 2/20 0.37
TUBA3E Q6PEY2 2/20 0.37
TUBA1A Q71U36 2/20 0.37
TUBA1C Q9BQE3 2/20 0.37
TUBB6 Q9BUF5 2/20 0.37
TUBB2B Q9BVA1 2/20 0.37
TUBB1 Q9H4B7 2/20 0.37
EGFR P00533 1/20 0.37
PDGFRB P09619 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6958549 0.86 DRD1 (0.44) DRD1DRD2DRD4TUBB4ATUBB
SCHEMBL6958205 0.85 DRD1 (0.37) DRD1KDM4EKMT2AALDH1A1
Hydrochloric Acid SCHEMBL6963712 0.80 CA1 (0.37) EGFRPDGFRBKDRCA1CA2
SCHEMBL6968163 0.78 DRD1 (0.39) DRD1DRD2TUBB4ATUBBTUBA3C
SCHEMBL6989000 0.73 DRD1 (0.39) DRD1SIGMAR1
SCHEMBL6160361 0.73 ESR1 (0.34)
SCHEMBL6159540 0.73 HTR2A (0.36) HTR2C
SCHEMBL5518952 0.70 DRD1 (0.51) DRD1DRD2DRD4CA1CA2
Hydrochloric Acid SCHEMBL6964992 0.69 CA1 (0.40) EGFRPDGFRBKDRCA1CA2
Hydrochloric Acid SCHEMBL6958005 0.69 KCNH3 (0.35) KDM4EKMT2AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015444-B1 PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORP LTD (KR) 2003-05-28 EP disclosed
US-6352993-B1 ANTIULCER AGENTS YUHAN CORPORATION (KR) 2002-03-05 US disclosed
EP-1015444-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION, LTD. (KR) 2000-07-05 EP disclosed
WO-1998043968-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 1998-10-08 WO disclosed