SCHEMBL6958205

SCHEMBL6958205

COCc1nc(Cl)nc(N2CCc3ccccc3C2C)c1C

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 2/20 0.37
LIPE Q05469 1/20 0.35
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
HPGD P15428 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PRMT5 O14744 1/20 0.33
SPR P35270 3/20 0.31
POLB P06746 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PRCP P42785 1/20 0.30
TRPM8 Q7Z2W7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6989000 0.88 DRD1 (0.39) DRD1LIPEMAPK1PRMT5SPR
SCHEMBL6969253 0.85 DRD1 (0.40) DRD1KDM4EALDH1A1KMT2A
SCHEMBL6957781 0.83 DRD1 (0.39) DRD1LIPEMAPK1SPRPRCP
SCHEMBL6995013 0.83 DRD1 (0.39) DRD1LIPEMAPK1SPRPRCP
SCHEMBL7000740 0.83 DRD1 (0.39) DRD1LIPEMAPK1SPRPRCP
Hydrochloric Acid SCHEMBL6958005 0.82 KCNH3 (0.35) KDM4EALDH1A1MEN1HPGDMAPK1
Hydrochloric Acid SCHEMBL6962670 0.80 MAP4K1 (0.35) KDM4EALDH1A1MEN1MAPK1KMT2A
Hydrochloric Acid SCHEMBL6965281 0.79 KCNH3 (0.40) KDM4EALDH1A1MEN1HPGDMAPK1
SCHEMBL6966656 0.77 CHRM3 (0.46) KDM4EALDH1A1MEN1HPGDHTT
Hydrochloric Acid SCHEMBL6967084 0.76 GALR2 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015444-B1 PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORP LTD (KR) 2003-05-28 EP disclosed
US-6352993-B1 ANTIULCER AGENTS YUHAN CORPORATION (KR) 2002-03-05 US disclosed
EP-1015444-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION, LTD. (KR) 2000-07-05 EP disclosed
WO-1998043968-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 1998-10-08 WO disclosed