SCHEMBL6159540

SCHEMBL6159540

Cc1nc(Cl)nc(N2CCc3cc(Cl)ccc3C2C)c1C

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
SRD5A1 P18405 4/20 0.33
SRD5A2 P31213 2/20 0.33
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32
NOTUM Q6P988 1/20 0.32
SLC6A15 Q9H2J7 1/20 0.31
TP53 P04637 1/20 0.30
ROCK1 Q13464 1/20 0.30
FKBP1A P62942 1/20 0.30
CXCR3 P49682 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6157859 0.90 HTR2A (0.37) HTR2AHTR2CHTR2BSRD5A1NOTUM
SCHEMBL6160361 0.88 ESR1 (0.34) SRD5A1NOTUM
SCHEMBL6958549 0.86 DRD1 (0.44) HTR2C
SCHEMBL7000740 0.85 DRD1 (0.39)
SCHEMBL6995013 0.85 DRD1 (0.39)
SCHEMBL6957781 0.85 DRD1 (0.39)
SCHEMBL6956621 0.83 MAOA (0.48)
SCHEMBL7833131 0.82 CDK9 (0.35) HTR2AFNTAFNTBTP53
SCHEMBL6157563 0.81 HTR2A (0.36) HTR2AHTR2C
Hydrochloric Acid SCHEMBL6160403 0.81 KCNH3 (0.36) HTR2AFNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131312-B1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORP LTD (KR) 2005-10-26 EP disclosed
CN-1159312-C Novel poyrimidine derivatives and process for preparation thereof ������������ʽ���� 2004-07-28 CN disclosed
US-6545008-B1 Inhibitory activity against gastric acid secretion YUHAN CORPORATION (KR) 2003-04-08 US disclosed
CN-1326453-A Novel poyrimidine derivatives and process for preparation thereof YUHAN CORP (KR) 2001-12-12 CN disclosed
EP-1131312-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION, LTD. (KR) 2001-09-12 EP disclosed
WO-2000029403-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 2000-05-25 WO disclosed