SCHEMBL6969463

SCHEMBL6969463

C=CCn1c(COC(N)=O)nc(C(C)C)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.32
KDM4E B2RXH2 2/20 0.32
HTT P42858 1/20 0.32
APLNR P35414 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
TSHR P16473 1/20 0.32
GAA P10253 2/20 0.31
LMNA P02545 2/20 0.31
GLA P06280 1/20 0.31
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
HSD17B10 Q99714 1/20 0.31
ANXA2 P07355 1/20 0.30
S100A10 P60903 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7080054 0.90 ALDH1A1 (0.31) ALDH1A1APLNRTDP1TSHR
SCHEMBL6969467 0.89 ALDH1A1 (0.35) ALDH1A1KDM4EAPLNRTDP1TSHR
SCHEMBL6961583 0.89 APLNR (0.31) ALDH1A1APLNRTDP1TSHR
SCHEMBL7083901 0.88 ALDH1A1 (0.35) ALDH1A1KDM4EHTTAPLNRTDP1
SCHEMBL6969155 0.88 LMNA (0.30) LMNA
SCHEMBL6965378 0.88 LMNA (0.32) ALDH1A1LMNA
SCHEMBL6967644 0.86 GLA (0.32) LMNAGLA
SCHEMBL6972388 0.86 CYP1A2 (0.30)
SCHEMBL6969451 0.86 MEN1 (0.38) ALDH1A1HTTLMNA
SCHEMBL6965572 0.85 CYP1A2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed