SCHEMBL6969468

SCHEMBL6969468

CC(C)c1nc(CNC(=O)C(F)(F)F)n(C)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.34
CHEK1 O14757 1/20 0.33
IKBKB O14920 1/20 0.33
DCLK1 O15075 1/20 0.33
ROCK2 O75116 1/20 0.33
RPS6KA5 O75582 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
PAK4 O96013 1/20 0.33
CHEK2 O96017 1/20 0.33
EGFR P00533 1/20 0.33
LCK P06239 1/20 0.33
PIM1 P11309 1/20 0.33
PHKG2 P15735 1/20 0.33
FER P16591 1/20 0.33
RPS6KB1 P23443 1/20 0.33
CDK2 P24941 1/20 0.33
MARK3 P27448 1/20 0.33
MAPK1 P28482 1/20 0.33
AKT1 P31749 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6965470 0.87 SETDB1 (0.33) HSP90B1
SCHEMBL6973791 0.86 CYP2C9 (0.33) HSP90B1
SCHEMBL6965682 0.85 TSHR (0.35) MAPTMAPK1ATMHSP90B1
SCHEMBL6967933 0.82 HSP90B1 (0.33) HSP90B1
SCHEMBL6960933 0.81 ALDH1A1 (0.30)
SCHEMBL6969352 0.81 HSP90B1 (0.31) HSP90B1
SCHEMBL6960253 0.80 PTGDR2 (0.32) HSP90B1
SCHEMBL8345413 0.79 ALDH1A1 (0.35) MAPTEGFRHSP90B1
SCHEMBL6961309 0.79 HSP90B1 (0.33) HSP90B1
SCHEMBL6961217 0.79 MALT1 (0.32) HSP90B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP claimed
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed