SCHEMBL6969984

SCHEMBL6969984

[CH2]NC(=O)c1cccc(I)c1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.51
HDAC2 Q92769 1/20 0.51
GRM5 P41594 1/20 0.51
F2 P00734 1/20 0.50
MTOR P42345 3/20 0.49
TP53BP1 Q12888 1/20 0.49
KAT6A Q92794 1/20 0.47
SIGMAR1 Q99720 1/20 0.43
MYC P01106 1/20 0.42
MAX P61244 1/20 0.42
KDM4E B2RXH2 2/20 0.41
EGLN2 Q96KS0 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
RAB9A P51151 1/20 0.41
HDAC6 Q9UBN7 3/20 0.40
HDAC8 Q9BY41 2/20 0.40
ALDH1A1 P00352 1/20 0.40
PKM P14618 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11524926 0.82 KDM4E (0.62) HDAC1HDAC2GRM5F2MTOR
SCHEMBL2293623 0.80 ALDH1A1 (0.63) HDAC1HDAC2GRM5F2MTOR
SCHEMBL2290042 0.80 HDAC8 (0.63) HDAC1HDAC2GRM5F2MTOR
SCHEMBL1926964 0.77 MTOR (0.52) HDAC1HDAC2GRM5F2MTOR
SCHEMBL3673898 0.77 KCNK3 (0.61) HDAC1HDAC2GRM5F2MEN1
SCHEMBL29532463 0.77 PARP1 (0.59) HDAC1HDAC2GRM5F2MTOR
SCHEMBL2093436 0.77 HDAC1 (0.44) HDAC1HDAC2GRM5F2MTOR
SCHEMBL1259478 0.77 PARP1 (0.59) HDAC1HDAC2GRM5F2MTOR
SCHEMBL3673834 0.76 ATM (0.58) HDAC1HDAC2GRM5F2MTOR
SCHEMBL18079795 0.76 CES2 (0.54) HDAC1HDAC2GRM5F2MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed