SCHEMBL6970942

SCHEMBL6970942

CC(C)c1nc(COCCOC(N)=O)n(Cc2ccccn2)c1Sc1cccc(Cl)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SLC6A9 P48067 3/20 0.34
ALDH1A1 P00352 1/20 0.33
PPP1CA P62136 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
TP53 P04637 2/20 0.33
ADRA1D P25100 1/20 0.33
GRM5 P41594 1/20 0.33
PKM P14618 2/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7081480 0.94 ADRA1D (0.34) MAPTNPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL6973416 0.93 MAPT (0.36) MAPTNPC1RAB9ASLC6A9ALDH1A1
SCHEMBL6965073 0.93 MAPT (0.35) MAPTNPC1RAB9ASLC6A9ALDH1A1
SCHEMBL7081501 0.93 NPC1 (0.38) MAPTNPC1RAB9ASLC6A9ALDH1A1
SCHEMBL6961282 0.91 SMN1; SMN2 (0.35) MAPTNPC1RAB9ASLC6A9ALDH1A1
SCHEMBL6967466 0.91 ALDH1A1 (0.33) NPC1RAB9AALDH1A1SMN1; SMN2TP53
SCHEMBL6969000 0.91 S1PR3 (0.36) NPC1RAB9ASLC6A9GRM5GRIN1
SCHEMBL6960270 0.89 ALDH1A1 (0.36) MAPTNPC1RAB9ASLC6A9ALDH1A1
SCHEMBL7080059 0.89 CFTR (0.38) MAPTNPC1RAB9AALDH1A1KMT2A
SCHEMBL6968857 0.88 PIM1 (0.33) SLC6A9KMT2ATP53GRM5KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed