SCHEMBL6970972

SCHEMBL6970972

Cc1ncccc1Cn1c(CCO)nc(C(C)C)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 1/20 0.31
P2RX7 Q99572 1/20 0.31
GABRA5 P31644 1/20 0.31
IL1B P01584 1/20 0.30
HSP90B1 P14625 1/20 0.30
TRAP1 Q12931 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7081079 0.94 HSP90B1 (0.33) HRH1HSP90B1TRAP1
SCHEMBL6966452 0.92 HRH1 (0.32) HRH1P2RX7GABRA5IL1BHSP90B1
SCHEMBL7087627 0.89 ENPP2 (0.31) GABRA5
SCHEMBL7081352 0.86 TDP1 (0.31) HSP90B1TRAP1
SCHEMBL6969765 0.85 SMN1; SMN2 (0.31)
SCHEMBL6969846 0.85 KDM4E (0.33) HSP90B1TRAP1
SCHEMBL7082531 0.85 HRH1 (0.34) HRH1HSP90B1TRAP1
SCHEMBL6965901 0.84 RAB9A (0.35)
SCHEMBL6975013 0.83 ENPP2 (0.30)
SCHEMBL6967282 0.83 TDP1 (0.32) GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed