SCHEMBL6971351

SCHEMBL6971351

N#Cc1c[c]ccc1Sc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.54
ALDH1A1 P00352 4/20 0.54
MAPT P10636 3/20 0.54
HPGD P15428 2/20 0.54
MAOA P21397 2/20 0.47
MAOB P27338 2/20 0.47
MCL1 Q07820 1/20 0.41
CYP1A2 P05177 6/20 0.40
CYP2C19 P33261 6/20 0.40
CYP2C9 P11712 5/20 0.40
CYP3A4 P08684 4/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CYP2D6 P10635 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ABCC9 O60706 1/20 0.36
ABCC8 Q09428 1/20 0.36
KCNJ11 Q14654 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29669365 0.79 KDM4E (0.62) KDM4EALDH1A1MAPTHPGDMAOA
SCHEMBL4011637 0.79 KDM4E (0.62) KDM4EALDH1A1MAPTHPGDMAOA
SCHEMBL1451915 0.79 MAOA (0.38) KDM4EALDH1A1MAPTHPGDMAOA
SCHEMBL11148751 0.74 L3MBTL1 (0.36) KDM4EALDH1A1MAPTHPGDMAOA
SCHEMBL6965981 0.73 MEN1 (0.31) ALDH1A1MEN1KMT2AARPOLB
SCHEMBL11461774 0.72 KDM4E (0.54) KDM4EALDH1A1MAPTHPGDMAOA
SCHEMBL408050 0.71 TSHR (0.33) KDM4EALDH1A1MAOAMAOBCYP1A2
SCHEMBL5218112 0.70 SIRT1 (0.38) KDM4EALDH1A1MAPTHPGDMAOA
SCHEMBL1691711 0.70 PDE7A (0.39) KDM4EALDH1A1MAPTHPGDMAOA
SCHEMBL9685487 0.70 MAOA (0.34) KDM4EALDH1A1MAPTHPGDMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed