SCHEMBL6971519

SCHEMBL6971519

COC(=O)c1ccc(N2CCN(CCCN3c4ccccc4CCc4ccccc43)CC2)nc1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.57
RAB9A P51151 1/20 0.57
KMT2A Q03164 1/20 0.57
DRD2 P14416 14/20 0.56
DRD4 P21917 14/20 0.56
DRD3 P35462 14/20 0.56
GRIN1 Q05586 1/20 0.53
GRIN2B Q13224 1/20 0.53
CHRM2 P08172 2/20 0.47
CHRM4 P08173 2/20 0.47
CHRM5 P08912 2/20 0.47
CHRM1 P11229 2/20 0.47
CHRM3 P20309 2/20 0.47
ADRB2 P07550 1/20 0.47
ADRB1 P08588 1/20 0.47
ADRA1D P25100 1/20 0.47
ADRA1A P35348 1/20 0.47
ADRA1B P35368 1/20 0.47
HRH1 P35367 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967413 0.88 DRD2 (0.63) DRD2DRD4DRD3GRIN1GRIN2B
Hydrochloric Acid SCHEMBL6972169 0.87 DRD2 (0.62) DRD2DRD4DRD3GRIN1GRIN2B
SCHEMBL6959989 0.81 DRD2 (0.60) DRD2DRD4DRD3GRIN1GRIN2B
SCHEMBL7087330 0.78 DRD2 (0.56) DRD2DRD4DRD3GRIN1GRIN2B
SCHEMBL1331652 0.77 RAB9A (0.73) NPC1RAB9AKMT2A
SCHEMBL7528163 0.76 KMT2A (0.68) NPC1RAB9AKMT2A
SCHEMBL9210414 0.76 KMT2A (0.72) NPC1RAB9AKMT2ACHRM4
SCHEMBL19581051 0.75 KMT2A (0.61) NPC1RAB9AKMT2ADRD2DRD4
SCHEMBL9203972 0.74 KMT2A (0.70) NPC1RAB9AKMT2ADRD2DRD4
SCHEMBL6964171 0.74 DRD3 (0.53) DRD2DRD4DRD3GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934312-B1 1,4-DISUBSTITUTED PIPERAZINES NOVO NORDISK AS (DK) 2003-03-19 EP disclosed
US-6133268-A 1,4-disubstituted piperazines NOVO NORDISK A/S (DK) 2000-10-17 US disclosed
US-6004961-A ANTIINFLAMMATORY AGENTS, ANALGESICS; NON-INSULIN-DEPENDENT DIABETES; AGE-RELATED OBESITY; DIBENZO(D,G)(1,3,6)DIOXAZOCINE DERIVATIVES NOVO NORDISK A/S (DK) 1999-12-21 US disclosed
EP-0934312-A1 1,4-DISUBSTITUTED PIPERAZINES NOVO NORDISK A/S (DK) 1999-08-11 EP disclosed
WO-1998015548-A1 1,4-DISUBSTITUTED PIPERAZINES NOVO NORDISK A/S (DK) 1998-04-16 WO disclosed