SCHEMBL6972081

SCHEMBL6972081

O=C1c2ccccc2CN1CCN1CCN(c2cccc(C(F)(F)F)n2)CC1

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 12/20 0.57
DRD2 P14416 7/20 0.57
DRD5 P21918 4/20 0.57
HTR1A P08908 2/20 0.53
HTR7 P34969 2/20 0.52
OPRM1 P35372 2/20 0.50
DRD1 P21728 4/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6712934 0.99 DRD3 (0.56) DRD3DRD2DRD5HTR1AHTR7
SCHEMBL6711558 0.83 DRD3 (0.56) DRD3DRD2DRD5HTR1AHTR7
SCHEMBL9725137 0.83 HTR1A (0.55) DRD3DRD2HTR1AHTR7OPRM1
SCHEMBL6711653 0.80 DRD3 (0.62) DRD3DRD2DRD5HTR1AHTR7
SCHEMBL6716162 0.79 DRD3 (0.69) DRD3DRD2DRD5HTR1AHTR7
SCHEMBL29799616 0.79 HTR1A (0.65) DRD3DRD2HTR1AHTR7OPRM1
SCHEMBL9725084 0.79 HTR1A (0.65) DRD3DRD2HTR1AHTR7OPRM1
SCHEMBL7082370 0.77 DRD3 (0.56) DRD3DRD2DRD5HTR1AHTR7
Hydrochloric Acid SCHEMBL6715836 0.77 DRD3 (0.55) DRD3DRD2DRD5HTR1AHTR7
Hydrochloric Acid SCHEMBL6719032 0.76 DRD3 (0.50) DRD3DRD2DRD5HTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296954-A1 BICYCLIC LACTAMS AND SULFONAMIDES WITH 5-HT1A-AFFINITY AND USE THEREOF FOR PREVENTING AND TREATING CEREBRAL ISCHAEMIA Abbott GmbH & Co. KG (DE) 2003-04-02 EP disclosed
WO-2002002529-A1 BICYCLIC LACTAMS AND SULFONAMIDES WITH 5-HT1A-AFFINITY AND USE THEREOF FOR PREVENTING AND TREATING CEREBRAL ISCHAEMIA ABBOTT GMBH & CO. KG (DE) 2002-01-10 WO disclosed