SCHEMBL6972484

SCHEMBL6972484

CC(C)c1c(Sc2cc(F)cc(F)c2)nc(COC(N)=O)n1Cc1ccncc1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 3/20 0.35
PIM1 P11309 1/20 0.33
PIM3 Q86V86 1/20 0.33
S1PR3 Q99500 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
TP53 P04637 1/20 0.31
POLB P06746 1/20 0.31
CYP19A1 P11511 1/20 0.31
TLR7 Q9NYK1 2/20 0.31
HPGD P15428 2/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CASP1 P29466 1/20 0.30
CASP7 P55210 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7081063 0.92 ENPP2 (0.35) ENPP2PIM1PIM3S1PR3TP53
SCHEMBL6972748 0.92 ENPP2 (0.35) ENPP2S1PR3MEN1KMT2ATP53
SCHEMBL6975044 0.92 ENPP2 (0.35) ENPP2S1PR3MEN1KMT2APOLB
SCHEMBL8113749 0.90 MEN1 (0.34) ENPP2PIM1PIM3S1PR3MEN1
SCHEMBL6962542 0.90 PIM1 (0.35) ENPP2PIM1PIM3S1PR3MEN1
SCHEMBL6973086 0.88 PIM1 (0.36) ENPP2PIM1PIM3S1PR3MEN1
SCHEMBL7084514 0.85 CSNK2A2 (0.37) PIM1PIM3S1PR3MEN1KMT2A
SCHEMBL6973926 0.85 LMNA (0.30)
SCHEMBL6961825 0.85 LMNA (0.30)
SCHEMBL6974519 0.85 ENPP2 (0.35) ENPP2PIM1PIM3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed