SCHEMBL7081063

SCHEMBL7081063

CC(C)c1c(Sc2cccc(F)c2)nc(COC(N)=O)n1Cc1ccncc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
PIM1 P11309 2/20 0.33
PIM3 Q86V86 1/20 0.33
S1PR3 Q99500 2/20 0.33
CA2 P00918 2/20 0.33
CA4 P22748 2/20 0.33
CYP3A4 P08684 3/20 0.33
CYP2D6 P10635 3/20 0.33
CYP2C9 P11712 3/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C19 P33261 2/20 0.33
EPHX1 P07099 1/20 0.32
USP2 O75604 2/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
MAPT P10636 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7078281 0.92 ENPP2 (0.36) ENPP2LMNATP53GRIN1GRIN2B
SCHEMBL6972484 0.92 ENPP2 (0.35) ENPP2TP53PIM1PIM3S1PR3
SCHEMBL7084514 0.90 CSNK2A2 (0.37) TP53PIM1PIM3S1PR3ALDH1A1
SCHEMBL6973086 0.89 PIM1 (0.36) ENPP2LMNATP53PIM1PIM3
SCHEMBL7080206 0.87 PDE4A (0.36) LMNAHPGDMAPTCDC7L3MBTL1
SCHEMBL7081810 0.87 CA2 (0.38) LMNAS1PR3CA2CA4EPHX1
SCHEMBL6973183 0.86 ENPP2 (0.35) ENPP2LMNATP53GRIN1GRIN2B
SCHEMBL8113749 0.85 MEN1 (0.34) ENPP2PIM1PIM3S1PR3ALDH1A1
SCHEMBL6962542 0.85 PIM1 (0.35) ENPP2LMNAPIM1PIM3S1PR3
SCHEMBL6975044 0.85 ENPP2 (0.35) ENPP2LMNAS1PR3ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed