SCHEMBL6972504

SCHEMBL6972504

CC(C)c1nc(C(O)CCCc2ccccc2)[nH]c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 4/20 0.33
OXER1 Q8TDS5 4/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MCL1 Q07820 1/20 0.32
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
FAAH O00519 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
PRCP P42785 1/20 0.31
CAPN1 P07384 1/20 0.31
TSSK1B Q9BXA7 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
GSK3B P49841 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973401 0.95 TDP1 (0.32) GPR84TDP1PRCPCAPN1
SCHEMBL6966853 0.89 TDP1 (0.33) TDP1CAPN1
SCHEMBL6965426 0.88 GPR84 (0.33) GPR84MCL1FAAHCAPN1TSSK1B
SCHEMBL7086339 0.85 TSHR (0.30)
SCHEMBL8508128 0.83 HSP90B1 (0.36)
SCHEMBL6961240 0.82 MAPK14 (0.34) GPR84CAPN1
SCHEMBL7078733 0.82 HSP90B1 (0.32)
SCHEMBL6973659 0.80 MEN1 (0.34) PRCPALDH1A1MAPT
SCHEMBL6975421 0.80 ADRB2 (0.38)
SCHEMBL6961954 0.80 HSP90B1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed