SCHEMBL6973401

SCHEMBL6973401

CC(C)c1nc(C(O)CCc2ccccc2)[nH]c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.32
SCN9A Q15858 2/20 0.31
ATM Q13315 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PRCP P42785 2/20 0.31
CAPN1 P07384 1/20 0.31
ADRB1 P08588 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31
GPR84 Q9NQS5 1/20 0.31
POLB P06746 1/20 0.30
FABP3 P05413 1/20 0.30
FABP4 P15090 1/20 0.30
FABP5 Q01469 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972504 0.95 GPR84 (0.33) TDP1PRCPCAPN1GPR84
SCHEMBL7086339 0.91 TSHR (0.30)
SCHEMBL6966853 0.90 TDP1 (0.33) TDP1CAPN1KMT2APOLBFABP3
SCHEMBL6961240 0.87 MAPK14 (0.34) CAPN1ADRB1KMT2AGPR84POLB
SCHEMBL8508128 0.84 HSP90B1 (0.36)
SCHEMBL7078733 0.83 HSP90B1 (0.32)
SCHEMBL6965426 0.82 GPR84 (0.33) CAPN1GPR84
SCHEMBL7081628 0.81 GPR84 (0.39) GPR84
SCHEMBL6973659 0.81 MEN1 (0.34) PRCPKMT2ACYP3A4CYP2D6SLC6A2
SCHEMBL6975421 0.81 ADRB2 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed