SCHEMBL6972660

SCHEMBL6972660

COC(=O)CCc1nc(C(C)C)c(Sc2cc(F)cc(F)c2)n1Cc1ccncc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 9/20 0.40
CYP11B1 P15538 2/20 0.38
CYP11B2 P19099 2/20 0.38
KDM4E B2RXH2 1/20 0.34
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
MAPK14 Q16539 2/20 0.33
P2RX3 P56373 1/20 0.33
MAPK13 O15264 1/20 0.33
MAPK12 P53778 1/20 0.33
MAPK11 Q15759 1/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
TBXA2R P21731 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6968454 0.92 ENPP2 (0.39) ENPP2CYP11B1CYP11B2KDM4ETP53
SCHEMBL6968985 0.90 KDM4E (0.38) ENPP2CYP11B1CYP11B2KDM4EP2RX3
SCHEMBL8343038 0.90 TBXA2R (0.42) ENPP2TBXA2R
SCHEMBL6968962 0.88 CYP11B1 (0.41) ENPP2CYP11B1CYP11B2KDM4ECCNC
SCHEMBL6968461 0.86 CYP11B1 (0.31) CYP11B1CYP11B2KDM4E
SCHEMBL7085356 0.86 ENPP2 (0.36) ENPP2MAPK14
SCHEMBL6969213 0.85 ENPP2 (0.35) ENPP2CYP11B1TP53POLBP2RX3
SCHEMBL6974458 0.85 S1PR3 (0.38) ENPP2KDM4E
SCHEMBL6967988 0.85 ENPP2 (0.35) ENPP2TP53POLBP2RX3
SCHEMBL7082084 0.84 ENPP2 (0.35) ENPP2TP53POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed