SCHEMBL6973128

SCHEMBL6973128

CC(=O)OC(C)c1nc(Sc2cccc(F)c2)c(C(C)C)[nH]1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TYMS P04818 1/20 0.35
SLC6A9 P48067 5/20 0.34
CA2 P00918 2/20 0.34
CA4 P22748 2/20 0.34
HAO1 Q9UJM8 1/20 0.33
LMNA P02545 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
ALDH1A1 P00352 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
XPO1 O14980 1/20 0.32
EPHX1 P07099 1/20 0.32
PIK3CA P42336 1/20 0.32
NOTUM Q6P988 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6961662 0.89 TYMS (0.31) TYMSLMNASMN1; SMN2
SCHEMBL7086270 0.88 CA2 (0.36) TYMSSLC6A9CA2CA4HAO1
SCHEMBL6964414 0.87 HPGD (0.38) TYMSSLC6A9LMNAALDH1A1
SCHEMBL6967036 0.86 LMNA (0.38) LMNASMN1; SMN2ALDH1A1
SCHEMBL7078284 0.83 ROCK1 (0.33) TYMSSLC6A9CA2CA4
SCHEMBL7084668 0.83 HSP90AA1 (0.38) LMNASMN1; SMN2ALDH1A1
SCHEMBL6961917 0.83 HAO1 (0.38) TYMSSLC6A9CA2CA4HAO1
SCHEMBL6962736 0.83 TYMS (0.35) TYMSSLC6A9CA2CA4HAO1
SCHEMBL6971303 0.82 HAO1 (0.33) TYMSSLC6A9CA2CA4HAO1
SCHEMBL6961646 0.80 TYMS (0.31) TYMSLMNASMN1; SMN2XPO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed