SCHEMBL6973342

SCHEMBL6973342

Nc1ccc(Cl)cc1C(=O)C1CCN(C(=O)c2ccccc2)CC1

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 15/20 0.67
MEN1 O00255 1/20 0.67
KMT2A Q03164 1/20 0.67
MAPT P10636 1/20 0.54
HSD11B1 P28845 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969906 0.84 MGLL (0.64) MGLLMEN1KMT2AHSD11B1
Hydrochloric Acid SCHEMBL6979800 0.83 MGLL (0.63) MGLLMEN1KMT2AHSD11B1
SCHEMBL6969303 0.82 POLB (0.60) MGLLHSD11B1
Hydrochloric Acid SCHEMBL6969837 0.81 POLB (0.59) MGLLHSD11B1
SCHEMBL1720910 0.80 MGLL (1.00) MGLLMEN1KMT2AMAPTHSD11B1
SCHEMBL6208966 0.80 MGLL (1.00) MGLLMEN1KMT2AMAPTHSD11B1
SCHEMBL30590434 0.80 RECQL (0.56) MGLLMEN1KMT2A
SCHEMBL2471282 0.80 RECQL (0.56) MGLLMEN1KMT2A
SCHEMBL11754253 0.79 HRH4 (0.54) MGLL
Hydrochloric Acid SCHEMBL9115524 0.78 RECQL (0.54) MGLLMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0892795-B1 PIPERIDINYLPYRAMIDINE DERIVATIVES SUMITOMO PHARMA (JP) 2003-01-08 EP disclosed
US-5948786-A BLOCKING TUMOR NECROSIS FACTOR SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1999-09-07 US disclosed
EP-0892795-A1 PIPERIDINYLPYRAMIDINE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1999-01-27 EP disclosed
WO-1997038992-A1 PIPERIDINYLPYRAMIDINE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1997-10-23 WO disclosed