SCHEMBL6973470

SCHEMBL6973470

CC(C)c1nc(CC#N)n(Cc2ccccn2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.33
HSP90B1 P14625 2/20 0.32
TRAP1 Q12931 2/20 0.32
ALDH1A1 P00352 3/20 0.32
AGTR1 P30556 1/20 0.32
NOX4 Q9NPH5 1/20 0.31
ALOX5AP P20292 1/20 0.31
P2RX3 P56373 1/20 0.31
ATM Q13315 1/20 0.31
AR P10275 1/20 0.31
KDM4E B2RXH2 1/20 0.30
GAA P10253 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
GRIN1 Q05586 1/20 0.30
GRIN2B Q13224 1/20 0.30
FKBP2 P26885 1/20 0.30
FKBP1A P62942 1/20 0.30
FKBP1B P68106 1/20 0.30
FKBP3 Q00688 1/20 0.30
FKBP4 Q02790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969433 0.93 KMT2A (0.38) PIK3CDALDH1A1AGTR1NOX4ALOX5AP
SCHEMBL7086006 0.89 ALOX5AP (0.33) PIK3CDALDH1A1ALOX5APATMAR
SCHEMBL6960816 0.89 S1PR3 (0.33) ALDH1A1ALOX5APATMARKDM4E
SCHEMBL6974447 0.87 MEN1 (0.34) PIK3CDHSP90B1TRAP1ALDH1A1AGTR1
SCHEMBL6976953 0.87 ALDH1A1 (0.33) HSP90B1TRAP1ALDH1A1AGTR1NOX4
SCHEMBL6975001 0.87 ALDH1A1 (0.33) PIK3CDHSP90B1TRAP1ALDH1A1AGTR1
SCHEMBL6969004 0.85 CYP1A2 (0.33) PIK3CDHSP90B1TRAP1ALDH1A1AGTR1
SCHEMBL7082531 0.85 HRH1 (0.34) HSP90B1TRAP1ALDH1A1AGTR1NOX4
SCHEMBL7082928 0.85 HRH1 (0.36) PIK3CDHSP90B1TRAP1ALDH1A1AGTR1
SCHEMBL6960568 0.85 GRIN1 (0.37) ALDH1A1NOX4ALOX5APATMAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed