SCHEMBL6976953

SCHEMBL6976953

CC(C)c1nc(CO)n(Cc2ccccn2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.33
AGTR1 P30556 1/20 0.33
HRH1 P35367 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
TP53 P04637 2/20 0.33
NOX4 Q9NPH5 1/20 0.32
ALOX5AP P20292 1/20 0.32
ADRA1D P25100 1/20 0.32
P2RX3 P56373 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HSP90B1 P14625 1/20 0.32
TRAP1 Q12931 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
TLR7 Q9NYK1 1/20 0.32
S1PR3 Q99500 2/20 0.31
GABRA1 P14867 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7079929 0.92 GRM5 (0.38) ALDH1A1AGTR1HRH1MEN1KMT2A
SCHEMBL7082531 0.92 HRH1 (0.34) ALDH1A1AGTR1HRH1MEN1KMT2A
SCHEMBL6970195 0.90 TLR7 (0.35) ALDH1A1AGTR1HRH1MEN1KMT2A
SCHEMBL6973657 0.90 HDAC1 (0.35) ALDH1A1HRH1MEN1KMT2ATP53
SCHEMBL6975001 0.90 ALDH1A1 (0.33) ALDH1A1AGTR1MEN1KMT2ATP53
SCHEMBL7081548 0.89 BRD4 (0.36) HRH1KMT2AALOX5APKDM4EGRIN1
SCHEMBL6968293 0.88 HSP90B1 (0.35) ALDH1A1MEN1KMT2ATP53KDM4E
SCHEMBL6963974 0.88 ALDH1A1 (0.37) ALDH1A1HRH1TP53ALOX5APKDM4E
SCHEMBL6969004 0.88 CYP1A2 (0.33) ALDH1A1AGTR1MEN1KMT2ATP53
SCHEMBL6974447 0.88 MEN1 (0.34) ALDH1A1AGTR1MEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed