SCHEMBL6969004

SCHEMBL6969004

CC(C)c1nc(CN(C)C)n(Cc2ccccn2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C19 P33261 2/20 0.33
TSHR P16473 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KDM4E B2RXH2 1/20 0.33
S1PR3 Q99500 1/20 0.33
ALDH1A1 P00352 2/20 0.32
AGTR1 P30556 1/20 0.32
GABRA1 P14867 2/20 0.32
GABRA5 P31644 2/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA3 P34903 1/20 0.32
GABRA2 P47869 1/20 0.32
NOX4 Q9NPH5 1/20 0.32
ALOX5AP P20292 1/20 0.32
P2RX3 P56373 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7079263 0.92 SLC6A2 (0.41) CYP1A2CYP2D6CYP2C19CYP3A4CYP2C9
SCHEMBL7083143 0.89 GABRA1 (0.34) CYP1A2CYP2D6CYP2C19TSHRS1PR3
SCHEMBL6973323 0.88 S1PR3 (0.34) KDM4ES1PR3ALDH1A1GABRA1GABRA5
SCHEMBL6976953 0.88 ALDH1A1 (0.33) KDM4ES1PR3ALDH1A1AGTR1GABRA1
SCHEMBL6975001 0.88 ALDH1A1 (0.33) TDP1ALDH1A1AGTR1GABRA1GABRA5
SCHEMBL6974447 0.86 MEN1 (0.34) TDP1KDM4ES1PR3ALDH1A1AGTR1
SCHEMBL7082928 0.86 HRH1 (0.36) CYP1A2CYP2C19KDM4ES1PR3ALDH1A1
SCHEMBL7082531 0.86 HRH1 (0.34) CYP1A2CYP2C19KDM4ES1PR3ALDH1A1
SCHEMBL6973470 0.85 PIK3CD (0.33) KDM4EALDH1A1AGTR1GABRA1GABRA5
SCHEMBL6970195 0.85 TLR7 (0.35) TDP1KDM4EALDH1A1AGTR1NOX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed