SCHEMBL6973506

SCHEMBL6973506

Cc1ccc(NC(=O)c2ccnc(Cl)c2)cc1NC(=O)c1cccc(CN2CCN(C)CC2)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.64
KIT P10721 13/20 0.56
CSF1R P07333 9/20 0.56
BRAF P15056 6/20 0.55
EGFR P00533 4/20 0.55
ABL1 P00519 5/20 0.54
BCR P11274 4/20 0.54
ABL2 P42684 2/20 0.54
PDGFRA P16234 2/20 0.54
PLK4 O00444 1/20 0.54
DDX3X O00571 1/20 0.54
GAK O14976 1/20 0.54
SLC22A2 O15244 1/20 0.54
MAPK13 O15264 1/20 0.54
CA12 O43570 1/20 0.54
SLC22A3 O75751 1/20 0.54
ABCB11 O95342 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
LMNA P02545 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7677867 0.91 HPGDS (0.66) HPGDSKITCSF1RBRAFEGFR
SCHEMBL7681667 0.90 HPGDS (0.63) HPGDSKITCSF1RBRAFEGFR
SCHEMBL6780729 0.88 HPGDS (0.67) HPGDSKITCSF1RBRAFEGFR
SCHEMBL6976773 0.88 HPGDS (0.67) HPGDSKITCSF1RBRAFEGFR
SCHEMBL6973537 0.87 HPGDS (0.62) HPGDSKITCSF1RBRAFEGFR
SCHEMBL6782706 0.87 HPGDS (0.75) HPGDSKITCSF1RBRAFEGFR
SCHEMBL6979840 0.86 HPGDS (0.61) HPGDSKITCSF1RBRAFEGFR
SCHEMBL6978632 0.86 BRAF (0.70) HPGDSKITCSF1RBRAFEGFR
SCHEMBL6968243 0.85 MAPK14 (0.61) HPGDSBRAFRAF1MAPK14
SCHEMBL6966564 0.85 HPGDS (0.65) HPGDSKITCSF1RBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115707-B1 BENZAMIDE DERIVATIVES AND THER USE AS CYTOKINE INHIBITORS ASTRAZENECA AB (SE) 2003-11-12 EP disclosed
US-6455520-B1 TUMOR NECROSIS FACTOR AND INTERLEUKIN INHIBITORS; ANTIINFLAMMATORY AGENTS, ANTIALLERGENS; BONE DISORDERS ASTRA ZENECA AB (SE) 2002-09-24 US disclosed
EP-1115707-A1 BENZAMIDE DERIVATIVES AND THER USE AS CYTOKINE INHIBITORS AstraZeneca AB (SE) 2001-07-18 EP disclosed
WO-2000018738-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS CYTOKINE INHIBITORS ASTRAZENECA AB (SE) 2000-04-06 WO disclosed