SCHEMBL6973511

SCHEMBL6973511

CC(C)c1nc(CO)n(Cc2ccccn2)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 11/20 0.36
GRIN1 Q05586 3/20 0.34
GRIN2B Q13224 3/20 0.34
HRH1 P35367 1/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
GFER P55789 1/20 0.33
ALOX5AP P20292 1/20 0.32
TLR9 Q9NR96 1/20 0.32
TLR8 Q9NR97 1/20 0.32
TLR7 Q9NYK1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967358 0.92 S1PR3 (0.35) S1PR3GRIN1GRIN2BHRH1ALDH1A1
SCHEMBL6967980 0.92 GRIN1 (0.39) S1PR3GRIN1GRIN2BALDH1A1KDM4E
SCHEMBL6973869 0.90 TLR7 (0.35) S1PR3GRIN1GRIN2BHRH1ALDH1A1
SCHEMBL7078209 0.90 S1PR3 (0.34) S1PR3GRIN1GRIN2BALDH1A1KDM4E
SCHEMBL7081548 0.89 BRD4 (0.36) GRIN1GRIN2BHRH1KDM4EALOX5AP
SCHEMBL6963974 0.88 ALDH1A1 (0.37) HRH1ALDH1A1KDM4ELMNAALOX5AP
SCHEMBL6960222 0.88 S1PR3 (0.36) S1PR3GRIN1GRIN2BTLR7
SCHEMBL6973323 0.88 S1PR3 (0.34) S1PR3GRIN1GRIN2BALDH1A1KDM4E
SCHEMBL6969106 0.88 HRH1 (0.36) S1PR3GRIN1GRIN2BHRH1ALOX5AP
SCHEMBL7081701 0.88 S1PR3 (0.34) S1PR3GRIN1GRIN2BHRH1TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed