SCHEMBL6973869

SCHEMBL6973869

CC(C)c1nc(CCCO)n(Cc2ccccn2)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 2/20 0.35
S1PR3 Q99500 10/20 0.34
HRH1 P35367 1/20 0.33
GRIN1 Q05586 2/20 0.32
GRIN2B Q13224 2/20 0.32
ALDH1A1 P00352 2/20 0.31
TDP1 Q9NUW8 1/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
GFER P55789 1/20 0.31
ALOX5AP P20292 1/20 0.31
TLR9 Q9NR96 1/20 0.31
TLR8 Q9NR97 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967358 0.94 S1PR3 (0.35) TLR7S1PR3HRH1GRIN1GRIN2B
SCHEMBL6974995 0.93 GRIN1 (0.36) TLR7S1PR3HRH1GRIN1GRIN2B
SCHEMBL6973511 0.90 S1PR3 (0.36) TLR7S1PR3HRH1GRIN1GRIN2B
SCHEMBL6974738 0.90 TLR7 (0.36) TLR7HRH1GRIN1GRIN2BALDH1A1
SCHEMBL7084830 0.89 TLR7 (0.40) TLR7HRH1ALDH1A1TDP1ALOX5AP
SCHEMBL6970195 0.89 TLR7 (0.35) TLR7HRH1ALDH1A1TDP1KDM4E
SCHEMBL6969106 0.89 HRH1 (0.36) TLR7S1PR3HRH1GRIN1GRIN2B
SCHEMBL8344784 0.87 LMNA (0.38) S1PR3ALDH1A1KDM4ELMNAGFER
SCHEMBL6973313 0.87 GRIN1 (0.38) TLR7S1PR3HRH1GRIN1GRIN2B
SCHEMBL7079248 0.86 TDP1 (0.37) TLR7ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed