SCHEMBL6974410

SCHEMBL6974410

CC(C)c1nc(CO)n(CCCc2ccncc2)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.36
SIGMAR1 Q99720 3/20 0.32
GSK3B P49841 2/20 0.31
CYP17A1 P05093 2/20 0.30
CYP21A2 P08686 2/20 0.30
CYP11B1 P15538 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974089 0.94 POLB (0.34) MAPK14CYP17A1CYP21A2CYP11B1
SCHEMBL6966608 0.93 MAPK14 (0.37) MAPK14SIGMAR1GSK3B
SCHEMBL7084584 0.92 MAPK14 (0.37) MAPK14SIGMAR1GSK3B
SCHEMBL6965421 0.91 POLB (0.38) MAPK14SIGMAR1
SCHEMBL6960983 0.88 ENPP2 (0.32)
SCHEMBL6961438 0.87 MAPK14 (0.34) MAPK14SIGMAR1GSK3B
SCHEMBL6964205 0.87 HRH1 (0.32) MAPK14CYP17A1CYP21A2CYP11B1
SCHEMBL7080027 0.85 MAPK14 (0.31) MAPK14CYP17A1CYP21A2CYP11B1
SCHEMBL7084040 0.85 LMNA (0.31) MAPK14GSK3B
SCHEMBL6961236 0.85 POLB (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed