SCHEMBL6974427

SCHEMBL6974427

CC(C)c1nc(COC(N)=O)n(CCc2ccccc2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.38
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
NPSR1 Q6W5P4 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
USP2 O75604 1/20 0.35
ALDH1A1 P00352 3/20 0.35
L3MBTL1 Q9Y468 3/20 0.35
HTT P42858 2/20 0.34
GAA P10253 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PLK1 P53350 1/20 0.33
THRB P10828 1/20 0.33
PIK3CD O00329 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7081608 0.95 LMNA (0.36) MAPTMEN1KMT2AALDH1A1TDP1
SCHEMBL6964425 0.92 THRB (0.32) MAPTTHRB
SCHEMBL6960609 0.92 MAPT (0.37) MAPTMEN1KMT2ANPSR1CYP3A4
SCHEMBL6967638 0.92 TDP1 (0.39) MAPTMEN1KMT2AALDH1A1L3MBTL1
SCHEMBL6973948 0.90 LMNA (0.42) MAPTMEN1KMT2ANPSR1CYP3A4
SCHEMBL6961071 0.89 ALDH1A1 (0.36) MAPTMEN1KMT2ANPSR1CYP3A4
SCHEMBL6972378 0.88 TP53 (0.35) MAPTMEN1KMT2ASMN1; SMN2THRB
SCHEMBL6972724 0.87 LMNA (0.40) MAPTMEN1KMT2ACYP3A4CYP2C9
SCHEMBL6967899 0.87 GLA (0.32)
SCHEMBL6972300 0.87 HSP90B1 (0.33) MAPTMEN1KMT2ANPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed