SCHEMBL6974958

SCHEMBL6974958

COc1cc(-c2ccccc2N)cc(OC)c1OC

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FYN P06241 8/20 0.55
ALDH1A1 P00352 5/20 0.50
TSHR P16473 2/20 0.50
TDP1 Q9NUW8 2/20 0.50
GAA P10253 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
ADRA2B P18089 1/20 0.50
PTGS1 P23219 1/20 0.50
BRD4 O60885 3/20 0.48
HSD17B10 Q99714 3/20 0.48
KDM4E B2RXH2 2/20 0.48
CYP3A4 P08684 1/20 0.47
ACHE P22303 1/20 0.47
HPGD P15428 1/20 0.46
BMPR1A P36894 1/20 0.46
TGFBR1 P36897 1/20 0.46
ACVRL1 P37023 1/20 0.46
ACVR1 Q04771 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29057290 0.86 FYN (0.49) FYNALDH1A1TSHRTDP1GAA
SCHEMBL395115 0.81 KIT (0.61) ALDH1A1TSHRTDP1GAASMN1; SMN2
SCHEMBL30610422 0.81 KIT (0.61) ALDH1A1TSHRTDP1GAASMN1; SMN2
SCHEMBL3788055 0.81 ALDH1A1 (0.68) ALDH1A1TSHRTDP1SMN1; SMN2ADRA2B
SCHEMBL16621433 0.81 ALDH1A1 (0.47) FYNALDH1A1TSHRTDP1GAA
SCHEMBL27880132 0.80 ALDH1A1 (0.48) FYNALDH1A1TSHRTDP1GAA
SCHEMBL29456755 0.80 KIT (0.44) ALDH1A1TSHRTDP1SMN1; SMN2ADRA2B
SCHEMBL13813534 0.79 ADORA3 (0.52) FYNALDH1A1BRD4HSD17B10KDM4E
SCHEMBL31607694 0.79 ALDH1A1 (0.47) FYNALDH1A1TSHRTDP1GAA
SCHEMBL13952628 0.79 TUBB4A (0.55) FYNALDH1A1GAACYP3A4ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0862560-B1 SUBSTITUTED 2-ANILINOPYRIMIDINES USEFUL AS PROTEIN KINASE INHIBITORS CELLTECH THERAPEUTICS LTD (GB) 2003-04-02 EP disclosed
US-6235746-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATIVE AGENT CELLTECH THERAPEUTICS, LIMITED (GB) 2001-05-22 US disclosed
US-5958935-A Substituted 2-anilinopyrimidines useful as protein kinase inhibitors CELLTECH THERAPEUTICS LIMITED (GB) 1999-09-28 US disclosed
EP-0862560-A1 SUBSTITUTED 2-ANILINOPYRIMIDINES USEFUL AS PROTEIN KINASE INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 1998-09-09 EP disclosed
WO-1997019065-A1 SUBSTITUTED 2-ANILINOPYRIMIDINES USEFUL AS PROTEIN KINASE INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 1997-05-29 WO disclosed