SCHEMBL6974980

SCHEMBL6974980

CC(C)c1c(Sc2ccccc2)nc(C=O)n1Cc1ccncc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
MAPT P10636 3/20 0.36
NPSR1 Q6W5P4 2/20 0.36
VDR P11473 1/20 0.36
HTT P42858 1/20 0.36
KDM4E B2RXH2 2/20 0.35
LMNA P02545 1/20 0.35
FLT1 P17948 1/20 0.34
KDR P35968 1/20 0.34
ALOX5AP P20292 1/20 0.34
S1PR3 Q99500 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
KMT2A Q03164 2/20 0.33
GSK3B P49841 1/20 0.33
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6965090 0.88 IDO1 (0.38) ALDH1A1MAPTVDRHTTKDM4E
SCHEMBL7082707 0.87 GRIN1 (0.38) ALDH1A1VDRHTTLMNAS1PR3
SCHEMBL6972397 0.87 KCNH2 (0.34) VDRHTTFLT1KDRS1PR3
SCHEMBL6971756 0.86 S1PR3 (0.32) VDRS1PR3KMT2AMEN1
SCHEMBL7081207 0.83 ALDH1A1 (0.40) ALDH1A1MAPTNPSR1VDRHTT
SCHEMBL6964826 0.82 VDR (0.36) ALDH1A1MAPTNPSR1VDRKDM4E
SCHEMBL6973406 0.81 KDM4E (0.36) ALDH1A1MAPTKDM4EFLT1KDR
SCHEMBL6973201 0.81 KDM4E (0.36) ALDH1A1MAPTKDM4EFLT1KDR
SCHEMBL7079123 0.77 MEN1 (0.37) ALDH1A1MAPTKDM4ES1PR3KMT2A
SCHEMBL6973949 0.76 MAPT (0.39) ALDH1A1MAPTNPSR1HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed