SCHEMBL697525

SCHEMBL697525

COC(=O)C1CC(S(=O)(=O)CC2CC2)CN1c1cc(C)nn1Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 1/20 0.43
SMYD3 Q9H7B4 2/20 0.40
ALDH1A1 P00352 2/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 1/20 0.39
KCNJ6 P48051 2/20 0.36
KCNJ5 P48544 2/20 0.36
KCNJ3 P48549 2/20 0.36
RAB9A P51151 2/20 0.36
GAA P10253 1/20 0.36
KMT2A Q03164 2/20 0.36
NPC1 O15118 1/20 0.36
CTSS P25774 1/20 0.35
FKBP1A P62942 1/20 0.35
USP30 Q70CQ3 1/20 0.35
CYP3A4 P08684 2/20 0.34
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL697523 1.00 AGTR2 (0.43) AGTR2SMYD3ALDH1A1MAPTHPGD
SCHEMBL697524 1.00 AGTR2 (0.43) AGTR2SMYD3ALDH1A1MAPTHPGD
SCHEMBL696518 0.92 ALDH1A1 (0.37) AGTR2SMYD3ALDH1A1MAPTHPGD
SCHEMBL2105222 0.92 ALDH1A1 (0.37) AGTR2SMYD3ALDH1A1MAPTHPGD
SCHEMBL695014 0.91 AGTR2 (0.49) AGTR2SMYD3KCNJ6KCNJ5KCNJ3
SCHEMBL695013 0.91 AGTR2 (0.49) AGTR2SMYD3KCNJ6KCNJ5KCNJ3
SCHEMBL696093 0.88 AGTR2 (0.46) AGTR2SMYD3ALDH1A1MAPTHPGD
SCHEMBL696094 0.88 AGTR2 (0.46) AGTR2SMYD3ALDH1A1MAPTHPGD
SCHEMBL696092 0.88 AGTR2 (0.46) AGTR2SMYD3ALDH1A1MAPTHPGD
SCHEMBL2106768 0.85 SMN1; SMN2 (0.35) ALDH1A1KCNJ6KCNJ5KCNJ3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP disclosed
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed