SCHEMBL6975437

SCHEMBL6975437

Nc1cc[c]c(Cc2cccc([N+](=O)[O-])c2)c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
TSHR P16473 2/20 0.49
CYP19A1 P11511 1/20 0.44
LMNA P02545 2/20 0.43
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MAPT P10636 2/20 0.40
SIGMAR1 Q99720 1/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
POLB P06746 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
PYCR1 P32322 1/20 0.39
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6979276 0.81 TSHR (0.53) ALDH1A1TSHRCYP19A1LMNACYP1A2
SCHEMBL3722491 0.78 RIPK1 (0.45) ALDH1A1TSHRCYP19A1LMNACYP1A2
SCHEMBL10918542 0.77 TSHR (0.71) ALDH1A1TSHRCYP19A1LMNACYP1A2
SCHEMBL6981018 0.75 MAOB (0.42) ALDH1A1CYP19A1MAPTSIGMAR1KDM4E
SCHEMBL6978567 0.74 ALDH1A1 (0.50) ALDH1A1SIGMAR1MEN1KMT2AMAOB
SCHEMBL6978736 0.74 TSHR (0.51) ALDH1A1TSHRCYP19A1LMNACYP1A2
SCHEMBL11286333 0.73 TSHR (0.45) ALDH1A1TSHRCYP19A1LMNACYP1A2
SCHEMBL6979279 0.73 TSHR (0.57) ALDH1A1TSHRCYP19A1LMNACYP1A2
SCHEMBL29864638 0.72 TSHR (0.65) ALDH1A1TSHRCYP19A1LMNACYP1A2
SCHEMBL5250015 0.72 TSHR (0.65) ALDH1A1TSHRCYP19A1LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343756-A2 1-ARYL- OR 1-ALKYLSULFONYL-HETEROCYCLYLBENZAZOLES AS 5-HYDROXYTRYPTAMINE-6 LIGANDS Wyeth (US) 2003-09-17 EP disclosed
WO-2002036562-A2 1-ARYL- OR 1-ALKYLSULFONYL-HETEROCYCLYLBENZAZOLES AS 5-HYDROXYTRYPTAMINE-6 LIGANDS WYETH (US) 2002-05-10 WO disclosed