SCHEMBL6976871

SCHEMBL6976871

N#Cc1ccc(CCC(=O)N2CCCc3cc(NCc4ccc5ccccc5c4)ccc32)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 2/20 0.49
TSHR P16473 2/20 0.46
ALDH1A1 P00352 2/20 0.46
MEN1 O00255 1/20 0.46
USP2 O75604 1/20 0.46
HPGD P15428 1/20 0.46
KMT2A Q03164 1/20 0.46
HSD17B10 Q99714 1/20 0.46
TP53 P04637 2/20 0.44
FPR1 P21462 2/20 0.42
FPR2 P25090 2/20 0.42
NR3C1 P04150 2/20 0.42
RAB9A P51151 2/20 0.41
NPC1 O15118 1/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MRGPRX4 Q96LA9 1/20 0.40
PARP1 P09874 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6976631 0.92 HSD17B3 (0.46) FFAR1TSHRALDH1A1MEN1USP2
SCHEMBL6979870 0.88 RAB9A (0.44) FFAR1TSHRALDH1A1MEN1USP2
SCHEMBL6985994 0.86 POLB (0.43) TSHRALDH1A1MEN1USP2HPGD
SCHEMBL6982160 0.85 NR3C1 (0.61) ALDH1A1MEN1KMT2ANR3C1MAPT
Hydrochloric Acid SCHEMBL7089726 0.85 FFAR1 (0.47) FFAR1ALDH1A1TP53NR3C1RAB9A
SCHEMBL6983653 0.84 FPR1 (0.44) TSHRALDH1A1MEN1USP2HPGD
SCHEMBL6981983 0.84 RAB9A (0.46) TSHRALDH1A1MEN1USP2HPGD
SCHEMBL6983538 0.83 FFAR1 (0.41) FFAR1TSHRALDH1A1MEN1USP2
SCHEMBL6986432 0.83 TP53 (0.48) TSHRALDH1A1MEN1USP2HPGD
SCHEMBL6986003 0.83 RAB9A (0.48) TSHRALDH1A1MEN1USP2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
US-6300342-B1 FOR THERAPY OR INHIBITING THROMBUS FORMATION; FOR THERAPY OF FIBRIN-DEPENDENT INFLAMMATORY CONDITION BOEHRINGER INGELHEIM PHARM KG (DE) 2001-10-09 US disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed