SCHEMBL6977407

SCHEMBL6977407

CC(C)CN(NC(=O)[C@H](CC1CCCC1)[C@H](CC=Cc1ccccc1)C(=O)NO)C(=O)[C@@H](C)N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 1/20 0.52
CTSC P53634 1/20 0.37
HTR2A P28223 3/20 0.36
MMP1 P03956 4/20 0.35
MMP2 P08253 4/20 0.35
MMP3 P08254 4/20 0.35
MMP8 P22894 4/20 0.35
MMP13 P45452 4/20 0.35
METAP2 P50579 1/20 0.34
METAP1 P53582 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
MASP2 O00187 1/20 0.34
GRIK1 P39086 2/20 0.33
GRIK2 Q13002 2/20 0.33
APP P05067 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983569 0.91 ADAM17 (0.48) ADAM17MMP1MMP2MMP3MMP8
SCHEMBL6986120 0.89 ADAM17 (0.48) ADAM17MMP1MMP2MMP3MMP8
SCHEMBL6981622 0.87 ADAM17 (0.68) ADAM17CTSCHTR2AMMP1MMP2
SCHEMBL6986009 0.86 ADAM17 (0.40) ADAM17CTSCHTR2AMETAP2METAP1
Hydrochloric Acid SCHEMBL6986451 0.86 ADAM17 (0.67) ADAM17CTSCHTR2AMMP1MMP2
SCHEMBL6988077 0.86 ADAM17 (0.39) ADAM17CTSCMETAP2METAP1
Hydrochloric Acid SCHEMBL6984718 0.80 ADAM17 (0.68) ADAM17CTSCHTR2AMMP1MMP2
Hydrochloric Acid SCHEMBL6986409 0.80 ADAM17 (0.68) ADAM17CTSCHTR2AMMP1MMP2
SCHEMBL6942318 0.79 ADAM17 (0.62) ADAM17MMP1MMP2MMP3MMP8
SCHEMBL6943944 0.79 ADAM17 (0.73) ADAM17MMP1MMP2MMP3MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1089964-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-10-29 EP disclosed
US-6239151-B1 TREATMENT OF INFLAMMATORY AND AUTOIMMUNE DISEASES, OSTEOARTHRITIS, RESPIRATORY DISEASES, TUMORS, CACHEXIA, CARDIOVASCULAR DISEASES, FEVER, HAEMORRHAGE AND SEPSIS, HYDRAZINE DERIVATIVES, HOFFMANN-LA ROCHE INC. 2001-05-29 US disclosed