SCHEMBL6977503

SCHEMBL6977503

COC(OCC[Si](C)(C)C)c1cccc(-c2cccn2C(=O)OC(C)(C)C)n1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.45
HSP90AB1 P08238 1/20 0.45
PIK3R1 P27986 1/20 0.38
PIK3CA P42336 1/20 0.38
ATR Q13535 1/20 0.34
TNK2 Q07912 1/20 0.34
TGFBR1 P36897 2/20 0.33
BUB1 O43683 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6977508 0.77 HSP90AA1 (0.45) HSP90AA1HSP90AB1PIK3R1PIK3CAATR
SCHEMBL22940781 0.74 HSP90AA1 (0.58) HSP90AA1HSP90AB1PIK3R1PIK3CAATR
SCHEMBL2786895 0.73 HSP90AA1 (0.63) HSP90AA1HSP90AB1PIK3R1PIK3CAATR
SCHEMBL30040550 0.73 HSP90AA1 (0.67) HSP90AA1HSP90AB1PIK3R1PIK3CAATR
SCHEMBL24696520 0.73 HSP90AA1 (0.67) HSP90AA1HSP90AB1PIK3R1PIK3CAATR
SCHEMBL6984258 0.70
SCHEMBL24696638 0.68 HSP90AA1 (0.56) HSP90AA1HSP90AB1PIK3R1PIK3CAATR
SCHEMBL6983802 0.67 L3MBTL1 (0.33)
SCHEMBL3835540 0.67 HSP90AA1 (0.42) HSP90AA1HSP90AB1PIK3R1PIK3CAATR
SCHEMBL21074037 0.66 HSP90AA1 (0.61) HSP90AA1HSP90AB1PIK3R1PIK3CAATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946546-B1 PYRIDIN-2-YL-METHYLAMINE DERIVATIVES, METHOD OF PREPARING AND APPLICATION AS MEDICINE PF MEDICAMENT (FR) 2003-06-25 EP disclosed
US-6020345-A Pyridin-2-yl-methylamine derivatives, method of preparing and application as medicine PIERRE FABRE MEDICAMENT (FR) 2000-02-01 US disclosed