SCHEMBL6978487

SCHEMBL6978487

O=C1CCC(c2ccc3c(c2)[N]C(=O)N3)CC1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 3/20 0.44
EPHX2 P34913 2/20 0.39
PDE4A P27815 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4C Q08493 2/20 0.38
PDE4D Q08499 2/20 0.38
HRH3 Q9Y5N1 1/20 0.34
IKBKE Q14164 1/20 0.33
TBK1 Q9UHD2 1/20 0.33
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
DGAT1 O75907 1/20 0.32
NOTUM Q6P988 3/20 0.31
DDB1 Q16531 1/20 0.31
CRBN Q96SW2 1/20 0.31
PPARG P37231 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL788535 0.85 QDPR (0.45) EPHX2DDB1CRBN
SCHEMBL3827824 0.84 EPHX2 (0.38) EPHX2IKBKETBK1PRMT5WDR77
SCHEMBL6982209 0.80 EPHX2 (0.36) EPHX2HRH3PRMT5WDR77NOTUM
SCHEMBL4301270 0.78 SLC18A3 (0.48) EPHX2HRH3
SCHEMBL6211091 0.77 EPHX2 (0.34) EPHX2HRH3PRMT5WDR77
SCHEMBL4311163 0.76 TLR9 (0.42) EPHX2HRH3
Hydrochloric Acid SCHEMBL5720133 0.76 HPGD (0.40) EPHX2HRH3DDB1CRBN
SCHEMBL2334055 0.75 EPHX2 (0.41) ESR2EPHX2PRMT5WDR77NOTUM
SCHEMBL6213577 0.73 CYP2C9 (0.43) HRH3
SCHEMBL6212043 0.73 EPHX2 (0.36) EPHX2PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1286975-A1 BICLYCLIC CYCLOHEXYLAMINES AND THEIR USE AS NMDA RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2003-03-05 EP disclosed
WO-2001092239-A1 BICICLIC CYCLOHEXYLAMINES AND THEIR USE AS NMDA RECEPTOR ANTOGONISTS WARNER-LAMBERT COMPANY (US) 2001-12-06 WO disclosed