SCHEMBL6978748

SCHEMBL6978748

COC(=O)CC(=O)c1ccc(-c2cccs2)s1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.60
KDM4E B2RXH2 5/20 0.60
LMNA P02545 2/20 0.60
GAA P10253 2/20 0.60
L3MBTL1 Q9Y468 2/20 0.60
MAPT P10636 2/20 0.60
GLA P06280 1/20 0.60
HDAC1 Q13547 1/20 0.59
NPC1 O15118 5/20 0.56
RAB9A P51151 4/20 0.56
HPGD P15428 2/20 0.55
HSD17B10 Q99714 2/20 0.55
TP53 P04637 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
MEN1 O00255 1/20 0.55
POLB P06746 1/20 0.55
NFKB1 P19838 1/20 0.55
MAPK1 P28482 1/20 0.55
CASP1 P29466 1/20 0.55
CASP7 P55210 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31055049 0.81 KDM4E (0.68) ALDH1A1KDM4ELMNAGAAL3MBTL1
SCHEMBL12887317 0.81 ALDH1A1 (0.68) ALDH1A1KDM4ELMNAGAAL3MBTL1
SCHEMBL15803999 0.81 ALDH1A1 (0.67) ALDH1A1KDM4ELMNAGAAL3MBTL1
SCHEMBL8571801 0.80 ALDH1A1 (0.66) ALDH1A1KDM4ELMNAGAAL3MBTL1
SCHEMBL13942802 0.80 ALDH1A1 (0.65) ALDH1A1KDM4ELMNAGAAL3MBTL1
SCHEMBL1143695 0.79 ERCC5 (0.61) ALDH1A1LMNAGAAL3MBTL1MAPT
SCHEMBL8572921 0.78 ALDH1A1 (0.63) ALDH1A1KDM4ELMNAGAAL3MBTL1
SCHEMBL13140626 0.77 ALDH1A1 (0.61) ALDH1A1KDM4ELMNAGAAL3MBTL1
SCHEMBL8571740 0.77 ALDH1A1 (0.61) ALDH1A1KDM4ELMNAGAAL3MBTL1
SCHEMBL11973061 0.77 HDAC1 (0.59) ALDH1A1KDM4ELMNAGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109560-B1 COMPOUNDS USEFUL AS AICARFT INHIBITORS AGOURON PHARMA (US) 2003-08-27 EP disclosed
US-6525050-B1 Inhibit the enzyme aminoimidazole carboxamide ribonucleotide formyl transferase; antiproliferative agents; antitumor, antiinflammatory, antipsoriatic, and/or immunosuppressive AGOURON PHARMACEUTICALS, INC. 2003-02-25 US disclosed
EP-1109560-A4 COMPOUNDS USEFUL AS AICARFT INHIBITORS AGOURON PHARMA (US) 2002-04-17 EP disclosed
EP-1109560-A1 COMPOUNDS USEFUL AS AICARFT INHIBITORS AGOURON PHARMACEUTICALS, INC. (US) 2001-06-27 EP disclosed
WO-2000013688-A1 COMPOUNDS USEFUL AS AICARFT INHIBITORS AGOURON PHARMACEUTICALS, INC. (US) 2000-03-16 WO disclosed