SCHEMBL6978885

SCHEMBL6978885

CNc1cc(N2CCN(C(=O)N3CCN(S(=O)(=O)c4ccc(C(F)(F)F)cc4)CC3)CC2)ncn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
KDM4E B2RXH2 2/20 0.54
MAPT P10636 2/20 0.54
HDAC3 O15379 2/20 0.48
HDAC4 P56524 2/20 0.48
HDAC1 Q13547 2/20 0.48
HDAC7 Q8WUI4 2/20 0.48
HDAC2 Q92769 2/20 0.48
HDAC10 Q969S8 2/20 0.48
HDAC11 Q96DB2 2/20 0.48
HDAC8 Q9BY41 2/20 0.48
HDAC6 Q9UBN7 2/20 0.48
HDAC9 Q9UKV0 2/20 0.48
HDAC5 Q9UQL6 2/20 0.48
F13A1 P00488 1/20 0.47
TGM2 P21980 1/20 0.47
TGM1 P22735 1/20 0.47
PDGFRB P09619 1/20 0.47
CCR6 P51684 1/20 0.46
HSD11B1 P28845 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6980671 0.88 CCR6 (0.51) ALDH1A1KDM4EMAPTCCR6L3MBTL1
SCHEMBL6981045 0.88 LSS (0.54) ALDH1A1KDM4EMAPTHDAC3HDAC4
SCHEMBL6977047 0.87 LSS (0.51) ALDH1A1KDM4EMAPTL3MBTL1LMNA
SCHEMBL6975446 0.85 KDM4E (0.53) ALDH1A1KDM4EMAPTHDAC3HDAC4
SCHEMBL26429307 0.80 ALDH1A1 (0.57) ALDH1A1KDM4EMAPTHDAC3HDAC4
SCHEMBL26429286 0.76 KDM4E (0.51) ALDH1A1KDM4EMAPTHDAC3HDAC4
SCHEMBL7085163 0.76 LSS (0.69) ALDH1A1F13A1TGM2TGM1L3MBTL1
SCHEMBL7442116 0.75 L3MBTL1 (0.58) ALDH1A1KDM4EHDAC3HDAC4HDAC1
SCHEMBL6967361 0.74 LSS (0.53) KDM4EMAPTLMNAGAA
SCHEMBL6970581 0.74 LSS (0.56) ALDH1A1KDM4EMAPTL3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0925286-B1 SUBSTITUTED PYRIMIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE ASTRAZENECA AB (SE) 2003-01-02 EP disclosed
EP-0925286-A1 SUBSTITUTED PYRIMIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE ZENECA LIMITED (GB) 1999-06-30 EP disclosed
WO-1998006705-A1 SUBSTITUTED PYRIMIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE ZENECA LIMITED (GB) 1998-02-19 WO disclosed