SCHEMBL6978896

SCHEMBL6978896

CN1CC(CO)Oc2cc(Cl)ccc21

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.47
NISCH Q9Y2I1 5/20 0.42
KLKB1 P03952 1/20 0.41
HRH4 Q9H3N8 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
PTGIR P43119 1/20 0.38
RORC P51449 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
THRB P10828 1/20 0.36
AR P10275 1/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
CASR P41180 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5645322 0.84 NISCH (0.50) NISCHPTGIRRORCLMNATP53
SCHEMBL6101300 0.82 HTR1A (0.44) HTR1ANISCHPTGIRARMAOA
SCHEMBL6097146 0.80 NISCH (0.44) NISCHHRH3PTGIRTP53THRB
SCHEMBL6102026 0.80 CASR (0.49) HTR1ANISCHPTGIRCASR
SCHEMBL731248 0.80 CASR (0.49) HTR1ANISCHPTGIRCASR
SCHEMBL1689633 0.80 CASR (0.49) HTR1ANISCHPTGIRCASR
SCHEMBL6098334 0.76 NISCH (0.48) NISCHPTGIRRORCLMNATP53
SCHEMBL7817626 0.76 NISCH (0.48) NISCHPTGIRRORCLMNATP53
SCHEMBL31378741 0.75 RORC (0.39) NISCHRORCTHRBMAOAMAOB
SCHEMBL6100304 0.75 NISCH (0.49) HTR1ANISCHPTGIRRORCLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140925-B1 (3,4 DIHYDRO-2H-BENZO[1,4] OXAZINYL-METHYL)- 3-(1H-INDOL-3- YL)-ALKYL -AMINES WYETH CORP (US) 2003-04-23 EP disclosed
CN-1335845-A 3,4-dihydro-2H-benzo[1,4] oxazinyl-methyl [3-(1H-indol-3-yl)-alkyl]-amines AMERICAN HOME PROD (US) 2002-02-13 CN disclosed
US-6313114-B1 ANTIDEPRESSANTS AMERICAN HOME PRODUCTS CORP 2001-11-06 US disclosed
EP-1140925-A1 (3,4 DIHYDRO-2H-BENZO[1,4] OXAZINYL-METHYL)- 3-(1H-INDOL-3- YL)-ALKYL -AMINES AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-10 EP disclosed
WO-2000040580-A1 3,4-DIHYDRO-2H-BENZO[1,4]OXAZINYL-METHYL[3-(1H-INDOL-3-YL)-ALKYL]-AMINES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-07-13 WO disclosed